Sciencemadness Discussion Board

Nitromethane synthesis from methylamine

Glass mycologist - 3-11-2020 at 13:31

Hi there
I tried to look online for the nitromethane synthesis from methylamine but it's not very popular.
I found that oxidation of primary amine to nitro compounds is done using ozone or peroxides but does anyone have a procedure involving more "common" reagent ?

BluBoirt - 3-11-2020 at 15:36

This could give you some starting point. But maybe using chloroacetic acid as a starting material would be better than MeNH2.

https://patents.google.com/patent/CN102190587A/en

[Edited on 3-11-2020 by BluBoirt]

Herr Haber - 3-11-2020 at 16:40

I looked that up a couple of months ago when people were talking about ozone as a disinfectant.
Oddly enough I discovered some research paper where they would further react the produced nitromethane with chlorine with obvious results.

Opylation - 9-11-2020 at 00:46

I was looking at a bunch of different resources a little bit ago for the preparation of nitroalkanes. This one looks like the best process that has detailed instructions http://www.orgsyn.org/demo.aspx?prep=CV1P0401

I was also looking at oxidation of amines as a route. Now the oxidation of plain amines is a little tedious as you have to work up to nitro through a few different oxidation states and it didn’t seem too straight forward. One process though that looks really intriguing is oxidation of alpha-amino acids and then subsequent decarboxylation. Alpha-nitro acids easily decarboxylate via a similar mechanism to beta-oxoacids. I also thing the carbonyl aids in oxidation or at least promotes it. Look into oxidation of glycine. Decarboxylating the nitroacid will be a breeze

[Edited on 9-11-2020 by Opylation]

njl - 9-11-2020 at 05:12

@Opylation I have also done some reading about amine --> nitro and I think going from amine to oxime and then oxidizing to nitro is a good method. I don't have a procedure or anything but if I recall correctly the oxidation of primary amines to oximes is fairly gentle.